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Sharma, R.; Gatchie, L.; Williams, I.S.; Jain, S. K.; Vishwakarma, R.A.; Chaudhuri, B.; Bharate, S. B. Glycyrrhiza glabra extract and quercetin reverses cisplatin resistance in triple-negative MDA-MB-468 breast cancer cells via inhibition of cytochrome P450 1B1 enzyme. Bioorganic & Medicinal Chemistry Letters ,2017, 27(24), 5400-5403. |
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Horley ,N. J.; Beresford, K.J .M; Kaduskar ,S.; McCann, G.J .P; Ruparelia, K.C; Sonawane ,V.R; Joshi, P.; Williams, I. S; Gatchie, L.; Bharate, S.B; et al. (E)-3-(3,4,5-Trimethoxyphenyl)-1-(pyridin-4-yl)prop-2-en-1-one, a heterocyclic chalcone is a potent and selective CYP1A1 inhibitor and cancer chemopreventive agent. Bioorganic & medicinal chemistry letters ,2017, 27(24), 5409-5414. |
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Jeelani, S.M.; Farooq, U.; Gupta, A.P.; Lattoo, S.K. Phytochemical evaluation of major bioactive compounds in different cytotypes of five species of Rumex L. Industrial Crops and Products ,2017, 109, 897-904. |
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Singh, U.; Chashoo, G.; Khan, S. U.; Mahajan, P.; Nargotra, A.; Mahajan, G.; Singh, A.; Sharma, A.; Mintoo, M.J.; Guru, S.K.; et al. Design of Novel 3-Pyrimidinylazaindole CDK2/9 Inhibitors with Potent In Vitro and In Vivo Antitumor Efficacy in a Triple-Negative Breast Cancer Model. Journal of Medicinal Chemistry ,2017, 60(23), 9470-9489. |
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Borgohain, H.; Devi, R.; Dheer, D.; Borah, B.J.; Shankar, R.; Das, S.K. Synthesis of Tetrahydroquinoline-Embedded Bridged Benzothiaoxazepine-1,1-dioxides. European Journal Of Organic Chemistry ,2017, (45), 6671-6679. |
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Rather, M.A.; Rasool, F.; Bhat, Z. S.; Dar, H.; Maqbool, M.; Amin, S.; Yousuf, S. K.; Ahmad, Z. Design and synthesis of indolopyridone hybrids as new antituberculosis agents. Microbial Pathogenesis ,2017, 113, 330-334. |
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Khan, S.; Kumar, A.; Gupta, R.; Ahmed, Q.N. The Ritter Reaction of 2-Oxoaldehydes at Room Temperature: Divergent Behaviour towards Acid Strength. ChemistrySelect ,2017, 2(34), 11336-11340. |
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Sharma, A.; Magotra, A.; Dogra, A.; Rath, S.K.; Rayees, S.; Wazir, P.; Sharma, S.; Sangwan, P.L.; Singh, S.; Singh, G.; Nandi, U. Pharmacokinetics, pharmacodynamics and safety profiling of IS01957, a preclinical candidate possessing dual activity against inflammation and nociception. Regulatory Toxicology and Pharmacology ,2017, 91, 216-225. |
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Arora, D.; Kumar, A.; Gupta, P.; Chashoo, G.; Jaglan, S. Preparation, characterization and cytotoxic evaluation of bovine serum albumin nanoparticles encapsulating 5-methylmellein: A secondary metabolite isolated from Xylaria psidii. Bioorganic & Medicinal Chemistry Letters ,2017, 27(23), 5126-5130. |
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Sharma, R.; Magotra, A.; Manhas, R.S.; Chaubey, A. Antagonistic potential of a psychrotrophic fungus: &ITTrichoderma velutinum&IT ACR-P1. Biological Control, 2017, 115, 12-17. |
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Kour, P.; Kumar, A.; Sharma, R.; Chib, R.; Khan, I.A.; Rai, V.K. Synthesis of 2-amino-4H-chromen-4-ylphosphonates and beta-phosphonomalonates via tandem Knoevenagel-Phospha-Michael reaction and antimicrobial. Research On Chemical Intermediates ,2017, 43(12), 7319-7329. |
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Alam, N.; Koul, M.; Mintoo, M.J.; Khare, V.; Gupta, R.; Rawat, N.; Sharma, P. R.; Singh, S. K.; Mondhe, D. M.; Gupta, P. N. Development and characterization of hyaluronic acid modified PLGA based nanoparticles for improved efficacy of cisplatin in solid tumor. Biomedicine & Pharmacotherapy ,2017, 95, 856-864. |
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Bhat, Z. S.; Rather, M.A.; Maqbool, M.; Ul Lah, H.; Yousuf, S. K.; Ahmad, Z. Cell wall: A versatile fountain of drug targets in Mycobacterium tuberculosis. Biomedicine & Pharmacotherapy ,2017, 95, 1520-1534. |
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Kaur ,M. S.; Kaur ,R.; Bhatia, R.; Kumar ,K.; Kaur, R.; Singh, V.; Shankar, R.; Rawal, R. K. Synthetic and medicinal perspective of thiazolidinones: A review. Bioorganic chemistry , 2017, 75406-423. |
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Singh, G.; Razak, M.; Katoch, M.; Singh, G.; Katoch ,A.; Goswami ,A.; Katoch, M.; Katoch ,A.; Goswami, A.; Kitchlu ,S. Bioactive and biocontrol potential of endophytic fungi associated with Brugmansia aurea Lagerh. FEMS microbiology letters ,2017, 364(21). |
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By Bhat, Z. S.; Rather, M. A.; Syed, K.Y.; Ahmad, Z. α-pyrones and their hydroxylated analogs as promising scaffolds against Mycobacterium tuberculosis. Future Medicinal Chemistry, 2017, 9(17), 2053-2067. |
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Kumar, C.; Rasool, R.U.; Iqra, Z.; Nalli, Y.; Dutt, P.; Satti, N.K.; Sharma, N.; Gandhi, S.G.; Goswami, A.; Ali, A. Alkyne-azide cycloaddition analogues of dehydrozingerone as potential anti-prostate cancer inhibitors via the PI3K/Akt/NF-kappa B pathway. MedChemComm, 2017, 8(11), 2115-2124. |
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Rather, M. A.; Lone, A.M.; Teli, B.; Bhat, Z. S.; Singh, P.; Maqbool, M.; Shairgojray, B. A.; Dar, M. J.; Amin, S.; Yousuf, S.K.; et al. The synthesis, biological evaluation and structure-activity relationship of 2-phenylaminomethylene-cyclohexane-1,3-diones as specific anti-tuberculosis agents. MedChemComm ,2017, 8(11), 2133-2141, DOI:10.1039/C7MD00350A. |
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Kumar, S.; Nalli, Y.; Qadri, M.; Riyaz-Ul-Hassan, S.; Satti, N. K.; Gupta, V.; Bhushan, S.; Ali, A. Isolation of three new metabolites and intervention of diazomethane led to separation of compound 1 & 2 from an endophytic fungus, Cryptosporiopsis sp. depicting cytotoxic activity. Medicinal Chemistry Research ,2017, 26(11), 2900-2908. |
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Wani, N. A.; Singh, G.; Shankar, S.; Sharma, A.; Katoch, M.; Rai, R. Short hybrid peptides incorporating β- and γ-amino acids as antimicrobial agents. Peptides ,2017, 97, 46-53. |
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Ayoob, I.; Lone, S.H.; Masood-ur-R.; Zargar, O.A.; Bashir, R.; Shakeel-u-R.; Khuroo, M.A.; Bhat, K.A. New Semi-Synthetic Rosmarinic Acid-Based Amide Derivatives as Effective Antioxidants. CHEMISTRYSELECT ,2017, 2(31), 10153-10156. |
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Rasool, F.; Nayak D.; Katoch, A.; Faheem, M. M.; Yousuf ,S. K.; Hussain, N.; Goswami ,A.; Mukherjee ,D.; Rasool, F.; Hussain ,N.; et al. Regiospecific Synthesis of Ring A Fused Withaferin A Isoxazoline Analogues: Induction of Premature Senescence by W-2b in Proliferating Cancer Cells. Scientific reports ,2017, 7(1), 13749. |
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Kumar, V.; Gupta, M.; Gandhi, S. G.; Bharate, S.S.; Kumar, A.; Vishwakarma, R. A.; Bharate, S. B. Anti-inflammatory chromone alkaloids and glycoside from Dysoxylum binectariferum. Tetrahedron Letters ,2017, 58(42), 3974-3978. |
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Singh, R.; Kumar, V.; Bharate, S. S.; Vishwakarma, R. A. Synthesis, pH dependent, plasma and enzymatic stability of bergenin prodrugs for potential use against rheumatoid arthritis. Bioorganic & Medicinal Chemistry ,2017, 25(20), 5513-5521. |
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Saneja, A.; Kumar, R.; Singh, A.; Dhar, D.R.; Mintoo, M. J.; Singh, G.; Mondhe, D. M.; Panda, A.K.; Gupta, P. N. Development and evaluation of long-circulating nanoparticles loaded with betulinic acid for improved anti-tumor efficacy. International Journal of Pharmaceutics (Amsterdam, Netherlands) ,2017, 531(1), 153-166. |
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Singh ,S.; Kalia ,N.P.; Khan ,I.A.; Singh, S.; Joshi, P.; Sharma ,P. R.; Kumar, A.; Bharate ,S. B.; Khan, I. A.; Joshi, P.; et al. Boeravinone B, A Novel Dual Inhibitor of NorA Bacterial Efflux Pump of Staphylococcus aureus and Human P-Glycoprotein, Reduces the Biofilm Formation and Intracellular Invasion of Bacteria. Frontiers in microbiology ,2017, 81868. |
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Rashid, S.; Bhat, B. A.; Mehta, G. Synthesis of pleurolactone and related mono- and sesquiterpenoids: Bioactive constituents of edible mushrooms. Tetrahedron Letters ,2017, 58(40), 3800-3802. |
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Sharma, R.; Abdullaha, M.; Bharate, S.B. Metal-Free Ionic-Liquid-Mediated Synthesis of Benzimidazoles and Quinazolin-4(3H)-ones from Benzylamines. Asian Journal of Organic Chemistry ,2017, 6(10), 1370-1374. |
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Shah, A.; Hassan, Q.P.; Mushtaq ,S.; Shah ,A. M.; Hussain ,A.; Shah ,A.; Hassan, Q. P.; Shah, A. M.; Hussain ,A. Chemoprofile and functional diversity of fungal and bacterial endophytes and role of ecofactors – A review. Journal of basic microbiology ,2017, 57(10), 814-826. |
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Chinthakindi, P.K.; Rath, S. K.; Singh, J.; Singh, S.; Koul, S.; Sangwan, P. L. Isolation of isoxanthanol and synthesis of novel derivatives as potential cytotoxic agents. Medicinal Chemistry Research ,2017, 26(10), 2499-2513. |
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Awasthi, P.; Singh, A.; Sheikh, G.; Mahajan, V.; Gupta, A.P.; Gupta, S.; Bedi, Y. S.; Gandhi, S. G. Mining and characterization of EST-SSR markers for Zingiber officinale Roscoe with transferability to other species of Zingiberaceae. Physiology and Molecular Biology of Plants ,2017, 23(4), 925-931. |
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Joshi, P.; Vishwakarma, R.A.; Bharate, S. B. Natural alkaloids as P-gp inhibitors for multidrug resistance reversal in cancer. European Journal of Medicinal Chemistry ,2017, 138, 273-292. |
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Jan ,A.T.; Rahman, S.; Yeo ,H.R.; Lee, E. J.; Choi ,I.; Malik ,M. A; Abdullah, T. S. Perspective Insights of Exosomes in Neurodegenerative Diseases: A Critical Appraisal. Frontiers in aging neuroscience ,2017,9317. |
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Sharma, S.; Kumar, A.; Mintoo ,M. J.; Mondhe, D. M.; Guru ,S. K.; Manda, S.; Bharate ,S. B. Prasad, V.D.; Sharma, P. R.; Bhushan ,S. A marine sponge alkaloid derivative 4-chloro fascaplysin inhibits tumor growth and VEGF mediated angiogenesis by disrupting PI3K/Akt/mTOR signaling cascade. Chemico-biological interactions,2017, 27547-60. |
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Sharma, R.; Abdullaha, M.; Bharate, S. B. Oxidant-Controlled C-sp2/sp3-H Cross-Dehydrogenative Coupling of N-Heterocycles with Benzylamines. Journal of Organic Chemistry ,2017, 82(18), 9786-9793. |
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Kumar, A.; Khan, S.; Ahmed, Q. N. Base-Controlled Reactions through an Aldol Intermediate Formed between 2-Oxoaldehydes and Malonate Half Esters. Organic Letters ,2017, 19(18), 4730-473. |
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Rasool, F.; Mukherjee, D. Pd-Catalyzed Regio- and Stereoselective C-Nucleoside Synthesis from Un-activated Uracils and Pyranoid Glycals. Organic Letters ,2017, 19(18), 4936-4939. |
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Singh ,H.; Singh ,J.V; Nepali, K.; Bedi, P. M. S; Gupta, M. K; Saxena, A. K; Sharma, S. Triazole tethered isatin-coumarin based molecular hybrids as novel antitubulin agents: Design, synthesis, biological investigation and docking studies. Bioorganic & medicinal chemistry letters ,2017, 27(17), 3974-3979. |
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Shah, A. M.; Shakeel,R.; Hussain, A.; Mushtaq, S.; Rather, M.A.; Shah, A.; Ahmad, Z.; Khan, I.A. ;Bhat, K.A.; Hassan, Q.P. Antimicrobial investigation of selected soil actinomycetes isolated from unexplored regions of Kashmir Himalayas, India. Microbial Pathogenesis ,2017, 110, 93-99. |
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Nissar, A. U.; Sharma, L.; Mudasir, M.A.; Nazir, L. A.; Umar, S. A.; Sharma, P.R.; Vishwakarma, R.A.; Tasduq, S. A. Chemical chaperone 4-phenyl butyric acid (4-PBA) reduces hepatocellular lipid accumulation and lipotoxicity through induction of autophagy. Journal of Lipid Research,2017, 58(9), 1855-186. |
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Pandith, S. A.; Dhar, N.; Wani, T.A.; Razdan, S.; Bhat, W. W.; Rana, S.; Khan, S.; Verma, M.K.; Lattoo, S.K. Production dynamics in relation to ontogenetic development and induction of genetic instability through in vitro approaches in Pelargonium graveolens: A potential essential oil crop of commercial significance. Flavour and Fragrance Journal,2017, 32(5), 376-387. |
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Hussain, A.; Rather, M. A.; Shah, A. M.; Bhat, Z. S.; Shah, A.; Ahmad, Z.; Parvaiz Hassan, Q. Antituberculotic activity of actinobacteria isolated from the rare habitats. Letters in Applied Microbiology ,2017, 65(3), 256-264. |
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Rather, S. A.; Shah, A.M.; Ali, S. A.; Dar, R. A.; Rah, B.; Ali, A.; Hassan, Q. P. Isolation and characterization of Streptomyces tauricus from Thajiwas glacier-a new source of actinomycin-D. Medicinal Chemistry Research ,2017, 26(9), 1897-1902. |
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Dar, N. J.; Bhat, J. A.; Satti, N. K.; Sharma, P. R.; Hamid, A.; Ahmad, M. Withanone, an Active Constituent from Withania somnifera, Affords Protection Against NMDA-Induced Excitotoxicity in Neuron-Like Cells. Molecular Neurobiology ,2017, 54(7), 5061-5073. |
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Williams, I. S.; Gatchie, L.; Chaudhuri ,B.; Williams, I. S.; Gatchie, L.; Chaudhuri, B.; Chib ,S.; Saran, S.; Nuthakki ,V.K.; Joshi ,P.; et al. Biotransformation of Chrysin to Baicalein: Selective C6-Hydroxylation of 5,7-Dihydroxyflavone Using Whole Yeast Cells Stably Expressing Human CYP1A1 Enzyme. Journal of agricultural and food chemistry ,2017, 65(34), 7440-7446. |
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Kour, G.; Singh, P. ; Bhagat, A.; Ahmed, Z. Biopharmaceutic parameters, pharmacokinetics, transport and CYP-mediated drug interactions of IIIM-017: A novel nitroimidazooxazole analogue with anti-tuberculosis activity. European Journal of Pharmaceutical Sciences ,2017,106, 71-78. |
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Husain ,I.; Bala ,K.; Wani, A.; Makhdoomi ,U.; Malik ,F.; Sharma, A. Arginase purified from endophytic Pseudomonas aeruginosa IH2: Induce apoptosis through both cell cycle arrest and MMP loss in human leukemic HL-60 cells. Chemico-biological interactions , 2017, 27435-49. |
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Wani, Z. A.; Sultan, P.; Ashraf, N.; Wani, Z. A.; Riyaz-Ul-Hassan ,S.; Ashraf, N.; Kumar, A.; Bindu ,K.; Riyaz-Ul-Hassan ,S. Mortierella alpina CS10E4, an oleaginous fungal endophyte of Crocus sativus L. enhances apocarotenoid biosynthesis and stress tolerance in the host plant. Scientific reports , 2017, 7(1), 8598. |
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Magotra, A.; Sharma, A.; Gupta, A. P.; Wazir, P.; Sharma, S.; Singh, P. P.; Tikoo, M.K.; Vishwakarma, R. A.; Singh, G.; Nandi, U. Development and validation of a highly sensitive LC-ESI-MS/MS method for estimation of IIIM-MCD-211, a novel nitrofuranyl methyl piperazine derivative with potential activity against tuberculosis: Application to drug development. Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences ,2017, 1060, 200-206. |
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Williams, I. S.; Gatchie, L.; Joshi, P.; Vishwakarma ,R.A.; Sharma, M.; Satti ,N. K.; Chaudhuri ,B.; Bharate ,S. B. Synthesis and biological evaluation of pyrrole-based chalcones as CYP1 enzyme inhibitors, for possible prevention of cancer and overcoming cisplatin resistance. Bioorganic & medicinal chemistry letters , 2017, 27(16), 3683-3687. |
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Gupta, L.; Sharma, A. K.; Gothwal ,A.; Khan, M. S.; Khinchi, M. P.; Qayum, A.; Singh, S.K.; Gupta ,U. Dendrimer encapsulated and conjugated delivery of berberine: A novel approach mitigating toxicity and improving in vivo pharmacokinetics. International journal of pharmaceutics ,2017, 528(1-2), 88-99. |
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Kumar, S.; Kour, G.; Schreckenbach, G.; Andotra, S.; Hundal, G.; Sharma, V.; Jaglan, S.; Pandey, S.K. 3,4-Dimethyl diphenyldithiophosphate of mononuclear cobalt(II) with N-donor ligands: Synthesis, structural characterization, DFT and antibacterial studies. Journal of Molecular Structure ,2017, 1141, 23-30. |
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Koul,M.; Kumar, A.; Singh, J.; Sharma ,P. R.; Singh ,S.; Koul, M.; Kumar ,A.; Deshidi ,R.; Sharma ,V.; Singh ,J.; et al. Cladosporol A triggers apoptosis sensitivity by ROS-mediated autophagic flux in human breast cancer cells. BMC cell biology ,2017, 18(1), 26. |
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Katoch, M.; Singh, G.; Paul, A.; Sridhar ,S .N. C. Fungal endophytes associated with Viola odorata Linn. as bioresource for pancreatic lipase inhibitors. BMC complementary and alternative medicine ,2017, 17(1), 385. |
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Mahajan, P.; Chashoo, G.; Gupta, M.; Kumar, A.; Singh, P. P.; Nargotra, A. Fusion of Structure and Ligand Based Methods for Identification of Novel CDK2 Inhibitors. Journal of Chemical Information and Modeling ,2017, 57(8), 1957-1969. |
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Khajuria, V.; Gupta, S.; Sharma, N.; Kumar, A.; Lone, N.A.; Khullar, M.; Dutt, P.; Sharma, P. R. Bhagat, A.; Ahmed, Z. Anti-inflammatory potential of hentriacontane in LPS stimulated RAW 264.7 cells and mice model. Biomedicine & Pharmacotherapy ,2017, 92, 175-186. |
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Batarseh ,Y.S; Kaddoumi ,A.; Bharate ,S.S.; Kumar, V.; Kumar, A.; Vishwakarma ,R. A.; Bharate ,S. B. Crocus sativus Extract Tightens the Blood-Brain Barrier, Reduces Amyloid β Load and Related Toxicity in 5XFAD Mice. ACS chemical neuroscience ,2017, 8(8), 1756-1766. |
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Katoch, M.; Singh, A.; Singh, G.; Wazir, P.; Kumar, R. Phylogeny, antimicrobial, antioxidant and enzyme-producing potential of fungal endophytes found in Viola odorata. Annals of Microbiology (Heidelberg, Germany) ,2017, 67(8), 529-540. |
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Gupta, N.; Rath, S. K.; Singh, J.; Qayum, A.; Singh, S.; Sangwan, P.L. Synthesis of novel benzylidene analogues of betulinic acid as potent cytotoxic agents. European Journal of Medicinal Chemistry , 2017, 135, 517-530. |
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Dheer, D.; Rawal, R. K.; Singh, V.; Sangwan, P. L.; Das, P.; Shankar, R. β-CD/CuI catalyzed regioselective synthesis of iodo substituted 1,2,3-triazoles, imidazo[1,2-a]-pyridines and benzoimidazo[2,1-b]thiazoles in water and their functionalization. Tetrahedron ,2017, 73(30), 4295-4306. |
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Gupta, N.; Sharma, S.; Raina, A.; Bhushan, S.; Malik, F. A.; Sangwan, P. L. Synthesis of Novel Mannich Derivatives of Bakuchiol as Apoptotic Inducer through Caspase Activation and PARP-1 Cleavage in A549 Cells. ChemistrySelect ,2017, 2(18), 5196-5201. |
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Nageswar, R. D.; Rasheed, S.k.; Raina, G.; Ahmed, Q. N.; Jaladanki, C. K.; Bharatam, P.V.; Das, P. Cobalt-catalyzed regioselective ortho C(sp2)-H bond nitration of aromatics through proton-coupled electron transfer assistance. Journal of Organic Chemistry ,2017, 82(14), 7234-7244. |
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Anil, K. K.; Kannaboina, P.; Das, P. Ruthenium-catalyzed site-selective C-H arylation of 2-pyridones and 1-isoquinolinones. Organic & Biomolecular Chemistry,2017, 15(26), 5457-5461. |
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Sharma, R.; Jamwal, V.; Singh, V. P.; Wazir, P.; Awasthi, P.; Singh, D.; Vishwakarma, R.A.; Gandhi, S.G.; Chaubey, Asha. Revelation and cloning of valinomycin synthetase genes in Streptomyces lavendulae ACR-DA1 and their expression analysis under different fermentation and elicitation conditions. Journal of Biotechnology, 2017, 253, 40-47. |
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Dar ,M.S.; Singh ,P.; Mir, R. A.; Dar ,M. J. Βeta-catenin N-terminal domain: An enigmatic region prone to cancer causing mutations. Mutation research , 2017, 773122-133. |
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Bhat, Z.S.; Rather, M.r A.; Maqbool, M.; Lah, H. U. L.; Yousuf, S. K.; Ahmad, Z.. α-pyrones: Small molecules with versatile structural diversity reflected in multiple pharmacological activities-an update. Biomedicine & Pharmacotherapy ,2017, 91, 265-277. |
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Singh, J.; Qayum, A.; Singh, R. D.; Koul, M.; Kaul, A.; Satti, N. K.; Dutt, P.; Hamid, A.; Singh, S. Immunostimulatory activity of plumieride an iridoid in augmenting immune system by targeting Th-1 pathway in balb/c mice. International Immunopharmacology ,2017, 48, 203-210. |
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Nayak, D.; Kumar, A.; Chakraborty, S.; Rasool, R.; Amin, H.; Katoch, A.; Gopinath, V.; Mahajan, V.; Zilla, M. K.; Rah, B.l; et al. Inhibition of Twist1-mediated invasion by Chk2 promotes premature senescence in p53-defective cancer cells. Cell Death & Differentiation ,2017, 24(7), 1275-1287. |
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Dangroo, N. A.; Singh, J.; Rath, S. K.; Gupta, N.; Qayum, A.; Singh, S.; Sangwan, P. L. A convergent synthesis of novel alkyne-azide cycloaddition congeners of betulinic acid as potent cytotoxic agent. Steroids , 2017, 123, 1-12. |
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Wadhwa, B.; Makhdoomi, U.; Vishwakarma ,R.; Malik, F. Protein kinase B: emerging mechanisms of isoform-specific regulation of cellular signaling in cancer. Anti-cancer drugs , 2017, 28(6), 569-580. |
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Ramaraju, P.; Mir, N.A.; Singh, D.; Sharma, P.; Kant, R.; Kumar, I. An Unprecedented Pseudo-[3+2] Annulation between N-(4-Methoxyphenyl)aldimines and Aqueous Glutaraldehyde: Direct Synthesis of Pyrrole-2,4-dialdehydes. European Journal of Organic Chemistry, 2017, (24), 3461-3465. |
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Wani, T.A.; Pandith, S. A.; Gupta, A. P.; Chandra, S.; Sharma, N.; Lattoo, S. K. Molecular and functional characterization of two isoforms of chalcone synthase and their expression analysis in relation to flavonoid constituents in Grewia asiatica L. PLoS One ,2017, 12(6), e0179155/1-e0179155/24. |
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Gupta, A.; Kaur, R.; Singh, D.; Kapoor, K.K. Graphene oxide: A carbocatalyst for the one-pot multicomponent synthesis of highly functionalized tetrahydropyridines. Tetrahedron Letters,2017, 58(26), 2583-2587. |
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Nalli, Y.; Thakur, V.; Mohmmed, A.; Gupta, V.K.; Ali, A. POCl3-mediated cyclization of (+)-S-mahanimbine led to the divergent synthesis of natural product derivatives with antiplasmodial activity. New Journal of Chemistry ,2017, 41(12), 4923-4930. |
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Mehra, R.; Khan, I. A.; Nargotra, A. Anti-tubercular drug discovery: in silico implications and challenges. European Journal of Pharmaceutical Sciences ,2017, 104, 1-15. |
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Hudwekar, A. D.; Reddy, G. L.; Verma, P. K.; Gupta, S.; Vishwakarma, R. A.; Sawant, S. D. Transition Metal-free Single Step Approach for Arylated Pyrazolopyrimidinones and Quinazolinones Using Benzylamines/Benzylalcohols/Benzaldehydes. ChemistrySelect ,2017, 2(17), 4963-4968. |
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Andotra ,S.; Kumar, S.; Kour ,M.; Chayawan, V.; Sharma ,V.; Jaglan ,S.; Pandey, S.K. Synthesis, spectroscopic, DFT and in vitro biological studies of vanadium(III) complexes of aryldithiocarbonates. Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy , 2017, 180127-137. |
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Guleria, S.; Singh, G.; Gupta, S.; Vyas, D. Antioxidant and oxidative DNA damage protective properties of leaf, bark and fruit extracts of Terminalia chebula. Indian Journal of Biochemistry & Biophysics, 2017, 54(4), 127-134. |
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Katoch, M.; Bindu, K.; Phull, S.; Verma, M. K. An endophytic Fusarium sp isolated from Monarda citriodora produces the industrially important plant-like volatile organic compound hexanal. Microbiology (London, United Kingdom) ,2017, 163(6), 840-847. |
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Joshi, P.; Gupta, M.; Vishwakarma, R. A.; Kumar, A.; Bharate, S. B. (Z)-2-(3-Chlorobenzylidene)-3,4-dihydro-N-(2-methoxyethyl)-3-oxo-2H-benzo[b][1,4]oxazine-6-carboxamide as GSK-3β inhibitor: Identification by virtual screening and its validation in enzyme- and cell-based assay. Chemical Biology & Drug Design ,2017, 89(6), 964-971. |
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Krishnan, A.; Abdullah, T.S.; Mounajjed, T.; Hartono, S.; McConico, A.; White, T.; LeBrasseur, N.; Lanza, I.; Nair, S.; Gores, G.; Charlton, M. A longitudinal study of whole body, tissue, and cellular physiology in a mouse model of fibrosing NASH with high fidelity to the human condition. American journal of physiology. Gastrointestinal and liver physiology ,2017, 312(6), G666-G680. |
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Joshi, P.; McCann, G.J. P.; Sonawane, V. R.; Vishwakarma, R. A.; Chaudhuri, B. Identification of Potent and Selective CYP1A1 Inhibitors via Combined Ligand and Structure-Based Virtual Screening and Their in Vitro Validation in Sacchrosomes and Live Human Cells. Journal of Chemical Information and Modeling ,2017, 57(6), 1309-1320, DOI:10.1021/acs.jcim.7b00095. |
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Hussain, A.; Rather, M. A.; Dar, M. S.; Aga, M. A.; Ahmad, N.; Manzoor, A.; Qayum, A.; Shah, A.; Mushtaq, S.; Ahmad, Z.; et al. Novel bioactive molecules from Lentzea violacea strain AS 08 using one strain-many compounds (OSMAC) approach. Bioorganic & Medicinal Chemistry Letters ,2017, 27(11), 2579-2582. |
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Malik, A. H.; Ashraf, N. Transcriptome wide identification, phylogenetic analysis, and expression profiling of zinc-finger transcription factors from Crocus sativus L. Molecular Genetics and Genomics ,2017, 292(3), 619-633. |
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Kumar, A.; Ahmed, Q.N. A Benzoquinone Imine Assisted Ring-Opening/Ring-Closing Strategy of the RCOCHN1N2 System: Dinitrogen Extrusion Reaction to Benzimidazoles. European Journal of Organic Chemistry ,2017, 2017(19), 2751-2756, DOI:10.1002/ejoc.201700357. |
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Das ,M.K.; Prajapati, B. K.; Ranjan ,K.; Tevatiya, S.; Sharma ,S.K.; Tiendrebeogo, R. W.; Kana, I. H.; Theisen, M.; Tiendrebeogo, R. W.; Kana ,I. H.; et al. Malaria epidemiology in an area of stable transmission in tribal population of Jharkhand, India. Malaria journal ,2017, 16(1), 181. |
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Rather, M.A.; Dar, B.A.; Shah, W.A.; Prabhakar, A.; Bindu, K.; Banday, J.A.; Qurishi, M.A. Comprehensive GC-FID, GC-MS and FT-IR spectroscopic analysis of the volatile aroma constituents of Artemisia indica and Artemisia vestita essential oils. Arabian Journal of Chemistry,2017, 10, S3798-S3803. |
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Rehman, S.; Latief, R.; Bhat, K.A.; Khuroo, M. A.; Shawl, A. S.; Chandra, S. Comparative analysis of the aroma chemicals of Melissa officinalis using hydrodistillation and HS-SPME techniques. Arabian Journal of Chemistry ,2017, 10(Suppl._2), S2485-S2490. |
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Rasool, R. U.; Nayak, D.; Chakraborty, S.; Faheem, M. M.; Rah, B.; Mahajan, P.; Gopinath, V.; Katoch, A.; Iqra, Z.; Yousuf, S. K.; et al. AKT is indispensable for coordinating Par-4/JNK cross talk in p21 downmodulation during ER stress. Oncogenesis ,2017, 6(5), e341. |
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Reddy, K. R.; Kannaboina, P.; Das, P. Palladium-Catalyzed Chemoselective Switch: Synthesis of a New Class of Indenochromenes and Pyrano[2,3-c]carbazoles. Asian Journal of Organic Chemistry ,2017, 6(5), 534-543. |
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Qadri, M.; Nalli, Y.; Jain, S. K.; Chaubey, A.; Ali, A.; Strobel, G.A.; Vishwakarma, R.A.; Riyaz-Ul-Hassan, S. An Insight into the Secondary Metabolism of Muscodor yucatanensis: Small-Molecule Epigenetic Modifiers Induce Expression of Secondary Metabolism-Related Genes and Production of New Metabolites in the Endophyte. Microbial Ecology ,2017, 73(4), 954-965. |
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Shah, A.; Rather, M. A.; Hassan, Q. P.; Aga, M. A.; Mushtaq, S.; Shah, A. M.; Hussain, A.; Baba, S. A.; Ahmad, Z. Discovery of anti-microbial and anti-tubercular molecules from Fusarium solani: an endophyte of Glycyrrhiza glabra. Journal of Applied Microbiology ,2017, 122(5), 1168-1176. |
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Ahmad, M.; Aga, M. A.; Bhat, J. A.; Kumar, B.; Rouf, A.; Capalash, N.; Mintoo, M.J.; Kumar, A.; Mahajan, P.; Mondhe, D. M.; et al. Exploring Derivatives of Quinazoline Alkaloid L-Vasicine as Cap Groups in the Design and Biological Mechanistic Evaluation of Novel Antitumor Histone Deacetylase Inhibitors. Journal of Medicinal Chemistry ,2017, 60(8), 3484-3497. |
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Siddique, M. ; Usman, M.; Jayaprakash ,V.; Sinha ,B. N.; McCann ,G. J .P.; Sonawane, V. R.; Horley, N.; Gatchie, L.; Joshi ,P.; Bharate ,S. B.; Chaudhuri, B. Quinazoline derivatives as selective CYP1B1 inhibitors. European journal of medicinal chemistry ,2017, 130320-327. |
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Ayoob, I.; Hazari, Y.M.; Lone, S.H.; Rehman ,S.; Khuroo, M.A.; Fazili, K.M.; Bhat, K.A. Phytochemical and Cytotoxic Evaluation of Peganum Harmala: Structure Activity Relationship Studies of Harmine. CHEMISTRYSELECT ,2017, 2(10), 2965-2968. |
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Singh, D.; Kumar, V.; Devi, N.; Malakar, C.C.; Shankar, R.; Singh, V. Metal-free Decarboxylative Amination: An Alternative Approach Towards Regioselective Synthesis of beta-Carboline N-fused Imidazoles. Advanced Synthesis & Catalysis,2017, 359(7), 1213-1226. |
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Thotakura, N.; Dadarwal, M.; Kumar ,P.; Raza, K.; Sharma ,G.; Katare ,O. P.; Guru, S. K.; Bhushan, S. Chitosan-Stearic Acid Based Polymeric Micelles for the Effective Delivery of Tamoxifen: Cytotoxic and Pharmacokinetic Evaluation. AAPS PharmSciTech ,2017, 18(3), 759-768. |
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Dheer ,D.; Singh ,V.; Shankar, R. Medicinal attributes of 1,2,3-triazoles: Current developments. Bioorganic chemistry ,2017, 7130-54. |
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Rather, L.J.; Akhter, S.; Padder, R.A.; Hassan, Q.P.; Hussain, M.; Khan, M.A.; Mohammad, F. Colorful and semi durable antioxidant finish of woolen yarn with tannin rich extract of Acacia nilotica natural dye. Dyes and Pigments,2017, 139, 812-819. |
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Saneja, A.; Sharma, L.; Singh, A.; Dubey, R. D.; Mintoo ,M.J.; Kumar, A.; Sangwan, P. L.; Abdullah, T. S.; Singh ,G,; Mondhe, D, M,; et al. Synthesis, characterization and augmented anticancer potential of PEG-betulinic acid conjugate. Materials science & engineering. C, Materials for biological applications ,2017, 73616-626. |
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Horley ,N. J.; Beresford ,K.J. M.; Chawla ,T.; McCann ,G. J. P.; Ruparelia, K.C; Sonawane ,V. R.; Tan, H. L.; Gatchie ,L.; Williams ,I. S.; Joshi, P.; et al. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines. European journal of medicinal chemistry ,2017, 129159-174. |
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Baba, S. A.; Vishwakarma, R.A.; Ashraf, N. Functional Characterization of CsBGlu12, a β-Glucosidase from Crocus sativus, Provides Insights into Its Role in Abiotic Stress through Accumulation of Antioxidant Flavonols. Journal of Biological Chemistry ,2017, 292(11), 4700-4713. |
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Katoch, M.; Phull ,S.; Vaid, S.; Singh ,S. uiversity, Phylogeny, anticancer and antimicrobial potential of fungal endophytes associated with Monarda citriodora L. BMC microbiology ,2017, 17(1), 44. |
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Ur Rasool, R.; Debasis, N.; Chakraborty, S.; Jamwal, V.L.; Mahajan, V.; Katoch, A.; Faheem, M. M..; Iqra, Z.; Amin, H.; Gandhi, S. G.; et al. Differential regulation of NM23-H1 under hypoxic and serum starvation conditions in metastatic cancer cells and its implication in EMT. European Journal of Cell Biology ,2017, 96(2), 164-171. |
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Dutta, S.; Godara ,R.; Katoch ,R.; Yadav ,A.; Katoch ,M.; Singh, N .K. Detection of amitraz and malathion resistance in field populations of Rhipicephalus (Boophilus) microplus (Acari: Ixodidae) in Jammu region of India. Experimental & applied acarology , 2017, 71(3), 291-301. |
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Singh, K.S.; Wang, P.; Narkhede, N.A.; Mozharivskyj, Y. Iridium(III) and Rhodium(III) compounds of dipyridyl-N-alkylimine and dipyridyl-NH-ketimine: Spectral characterization and crystal structure. Journal of Chemical Sciences ,2017, 129(3), 365-372. |
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Singh ,A.; Arvinda, S.; Suri ,J.; Singh ,S.; Koul, S.; Vishwakarma ,R.; Mondhe ,D. M.; Singh, G. IN0523 (Urs-12-ene-3α,24β-diol) a plant based derivative of boswellic acid protect Cisplatin induced urogenital toxicity. Toxicology and applied pharmacology , 2017, 3188-15. |
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Kumar, A.; Sharma, P. R.; Mondhe, D. M. Potential anticancer role of colchicine-based derivatives: an overview. Anti-Cancer Drugs ,2017, 28(3), 250-262. |
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Gurmeen, R.; Gobind, R.; Kaur, T.; Vyas, D.; Sharma, A. D.; Singh, J. Molecular cloning, characterization, heterologous expression and in-silico analysis of disordered boiling soluble stress-responsive wBsSRP protein from drought tolerant wheat cv.PBW 175. Plant physiology and biochemistry : PPB , 2017, 11229-44. |
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Magotra, A.; Kumar, M.; Kushwaha, M.; Awasthi, P.; Raina, C.; Gupta, A. P.; Shah, B. A.; Gandhi, S. G.; Chaubey, Asha. Epigenetic modifier induced enhancement of fumiquinazoline C production in Aspergillus fumigatus (GA-L7): an endophytic fungus from Grewia asiatica L. AMB Express , 2017, 7(1), 1-10. |
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Aga, M. A.; Rayees, S.; Rouf, A.; Kumar, B.; Sharma, A.; Nagaraju, P. V. V. S.; Singh, G.; Taneja, S.C. Synthesis of Ofornine mimics from natural product l-vasicine as anti-hypertensive agents. Bioorganic & Medicinal Chemistry ,2017, 25(4), 1440-1447. |
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Singh, G.; Singh ,G.; Bhatti ,R.; Gupta, V.; Mahajan ,A.; Singh, P.; Singh, I.M. P. Rationally designed benzopyran fused isoxazolidines and derived β(2,3,3)-amino alcohols as potent analgesics: Synthesis, biological evaluation and molecular docking analysis. European journal of medicinal chemistry ,2017, 127210-222. |
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Chinthakindi, P.K.; Singh, J.; Gupta, S.; Nargotra, A.; Mahajan, P.; Kaul, A.; Ahmed, Z.; Koul, S.; Sangwan, P.L. Synthesis of a-santonin derivatives for diminutive effect on T and B-cell proliferation and their structure activity relationships. European Journal of Medicinal Chemistry , 2017, 127, 1047-1058. |
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Gopalakrishna, P.;Geetha, K.; Bharate ,S.S.; Vishwakarma, R. A.; Awasthi ,A.; Verma ,R.; Mishra, G.; Singh, A. T.; Jaggi, M.; Mithal ,A. Antidiabetic potential of polyherbal formulation DB14201: Preclinical development, safety and efficacy studies. Journal of ethnopharmacology ,2017, 197218-230. |
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Devi ,P.; Wahidullah ,S.; Sheikh, F.; Pereira, R.; Amonkar, D.; Tilvi ,S.; Meena, R. M.; Narkhede Niteen. Biotransformation and Detoxification of Xylidine Orange Dye Using Immobilized Cells of Marine-Derived Lysinibacillus sphaericus D3. Marine drugs ,2017, 15(2). |
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Khan ,M. F.; Alam ,M. M.; Verma, G.; Akhtar, W.; Akhter ,M.; Shaquiquzzaman, M.; Rizvi ,M. A.; Ali, A. Molecular interactions of dioxins and DLCs with the ketosteroid receptors: an in silico risk assessment approach. Toxicology mechanisms and methods ,2017, 27(2), 151-163. |
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Dhamale, O.P.; Lawrence, R.; Wiegmann, E.M.; Shah, B.A.; Al-Mafraji, K.; Lamanna, W.C.; Lubke, T.; Dierks, T.; Boons, G.J.; Esko, J.D. Arylsulfatase K is the Lysosomal 2-Sulfoglucuronate Sulfatase. ACS Chemical Biology, 2017, 12(2), 367-373. |
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Rahat, B.; Kaur ,J.; Najar ,R.A.; Hamid, A.; Bagga ,R. The role of aberrant methylation of trophoblastic stem cell origin in the pathogenesis and diagnosis of placental disorders. Prenatal diagnosis ,2017, 37(2), 133-143. |
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Masood, R.; Mohammad ,Y.; Fazili ,K. M.; Bhat, K. A.; Ara, T. Synthesis and biological evaluation of novel 3-O-tethered triazoles of diosgenin as potent antiproliferative agents. Steroids , 2017, 1181-8. |
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Yedukondalu, N.; Arora, P.; Wadhwa, B.; Malik, F.A.; Vishwakarma, R.A.; Gupta, V. K.; Riyaz-Ul-Hassan, S.; Ali, A. Diapolic acid A-B from an endophytic fungus, Diaporthe terebinthifolii depicting antimicrobial and cytotoxic activity. Journal of Antibiotics ,2017, 70(2), 212-215. |
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121 |
Reddy, A. S.; Ranjith ,R.K.; Nageswar, R. D.; Jaladanki, C.K.; Bharatam, P.; Lam, P. Y. S.; Das, P. Copper(II)-catalyzed Chan-Lam cross-coupling: chemoselective N-arylation of aminophenols. Organic & Biomolecular Chemistry ,2017, 15(4), 801-806. |
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122 |
Mubashir, K.; Ganai, B. A.; Tantry, M.; Ghazanfar ,K.; Akbar, S.; Rah, B.; Masood, A. Anti-inflammatory and immuno-modulatory studies on LC-MS characterised methanol extract of Gentiana kurroo Royle. BMC complementary and alternative medicine ,2017, 17(1), 78. |
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123 |
Ravi ,C.; Chandra, M. D.; Qayum, A.; Singh ,S. K; Adimurthy ,S. Design, synthesis and cytotoxicity studies of novel pyrazolo[1, 5-a] pyridine derivatives. European journal of medicinal chemistry ,2017, 126277-285. |
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124 |
Yadav ,P.; Lal, K.; Kumar, A.; Guru, S. K.; Jaglan ,S.; Bhushan, S. Green synthesis and anticancer potential of chalcone linked-1,2,3-triazoles. European journal of medicinal chemistry ,2017, 126944-953. |
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125 |
Aruri, H.; Singh, U.; Kumar, M.; Sharma, S.; Aithagani, S. K.; Gupta, V. K.; Mignani, S.e; Vishwakarma, R.A.; Singh, P. Pal. Metal-free Cross-Dehydrogenative Coupling of HN-azoles with α-C(sp3)-H Amides via C-H Activation and Its Mechanistic and Application Studies. Journal of Organic Chemistry ,2017, 82(2), 1000-1012. |
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126 |
Rahat, B.; Mahajan ,A.; Kaur ,J.; Bagga ,R.; Hamid, A. Epigenetic modifications at DMRs of placental genes are subjected to variations in normal gestation, pathological conditions and folate supplementation. Scientific reports ,2017, 740774. |
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127 |
Borkar, S.R.; Bokolia, N.; Aidhen, I.S.; Khan, I.A. Synthesis of threo- and erythro-configured trihydroxy open chain lipophilic ketones as possible anti-mycobacterial agents. Tetrahedron-Asymmetry ,2017, 28(1). |
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128 |
Saneja, A.; Nayak ,D.; Srinivas, M.; Kumar ,A.; Khare, V.; Katoch ,A.; Goswami ,A.; Vishwakarma ,R. A; Sawant ,S. D.; Gupta, P. N. Development and mechanistic insight into enhanced cytotoxic potential of hyaluronic acid conjugated nanoparticles in CD44 overexpressing cancer cells. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences ,2017, 9779-91. |
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129 |
Dash, A.K.; Madhubabu, T.; Yousuf, S. K.; Raina, S.; Mukherjee, D. One-pot Mukaiyama type carbon-Ferrier rearrangement of glycals: Application in the synthesis of chromanone 3-C-glycosides. Carbohydrate Research ,2017, 438, 1-8. |
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130 |
Deshidi, R.; Devari, S.; Kushwaha, M.; Gupta, A.P.; Sharma, R.; Chib, R.; Khan, I.A.; Jaglan, S.; Shah, B.A. Isolation and Quantification of Alternariols from Endophytic Fungus, Alternaria alternata: LC-ESI-MS/MS Analysis. Chemistryselect ,2017, 2(1), 364-368. |
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131 |
Kour, M.; Kumar, S.; Andotra, S.; Kour, G.; Singh, G.; Gupta, V.K.; Kant, R.; Katoch, M.; Pandey, S.K. Chromium(III) complexes of dimethyl diphenyldithiophosphates: Synthesis, characterization, and antibacterial studies. Phosphorus Sulfur and Silicon and the Related Elements,2017, 192(10), 1119-1123. |
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132 |
Sharma, R; Khan, I. A. Mechanism and Potential Inhibitors of GlmU: A Novel Target for Antimicrobial Drug Discovery. Current Drug Targets ,2017,18(14), 1587-1597. |
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133 |
Dheer, D.; Reddy, K.R.; Rath, S.K.; Sangwan, P.L.; Das, P.; Shankar, R. Cu(I)-catalyzed double C-H amination: synthesis of 2-iodo-imidazo[1,2-a]pyridines . RSC Advances,2017, 7(64), 40591-40591. |
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134 |
Theisen ,M.; Adu, B.; Mordmuller, B.; Singh ,S. The GMZ2 malaria vaccine: from concept to efficacy in humans. Expert review of vaccines ,2017, 16(9), 907-917. |
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135 |
Nalli, Y.; Gupta, S.; Khajuria, V.; Singh, V. P.; Sajgotra, M.; Ahmed, Z.; Thakur, N. L.; Ali, A. TNF-α and IL-6 inhibitory effects of cyclic dipeptides isolated from marine bacteria Streptomyces sp. Medicinal Chemistry Research ,2017, 26(1), 93-100, DOI:10.1007/s00044-016-1730-8. |
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136 |
Valdiani, A.; Maziah ,M.; Abiri, R.; Talei, D.; Lattoo, S.r K.; Ortiz, R.; Rasmussen ,S.K.; Batley Jacqueline; Rafii Mohd Yusop; Maziah Mahmood; et al. Genoproteomics-assisted improvement of Andrographis paniculata: toward a promising molecular and conventional breeding platform for autogamous plants affecting the pharmaceutical industry. Critical reviews in biotechnology ,2017, 37(6), 803-816. |
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137 |
Khera, H.K.; Singh, S. K.; Mir, R.; Bharadwaj, V.; Singh, S. A HR-MS Based Method for the Determination of Chorismate Synthase Activity. Protein & Peptide Letters ,2017, 24(3), 229-234. |
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138 |
Katoch, M.; Pull ,S. Endophytic fungi associated with Monarda citriodora, an aromatic and medicinal plant and their biocontrol potential. Pharmaceutical biology ,2017, 55(1), 1528-1535. |
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139 |
Khare, V.; Al Sakarchi, W.; Gupta, P.N.; Curtis, A.D.M.; Hoskins, C. Synthesis and characterization of TPGS-gemcitabine prodrug micelles for pancreatic cancer therapy. RSC Advances,2017, 7(28), 17367-17367. |
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140 |
Sharma, S.; Gupta, M.K.; Saxena, A.K.; Bedi, P.M.S. Thiazolidinone Constraint Combretastatin Analogs as Novel Antitubulin Agents: Design, Synthesis, Biological Evaluation and Docking Studies. Anti-Cancer Agents in Medicinal Chemistry ,2017, 17(2), 230-240. |
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141 |
Shukla ,G.; Khare, P.; Patidar, R.; Saxena ,R.; Khera ,H. K.; Srivastava ,A. K. Therapeutic Potential, Challenges and Future Perspective of Cancer Stem Cells in Translational Oncology: A Critical Review. Current stem cell research & therapy ,2017, 12(3), 207-224. |
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142 |
Dheer,D.; Arora, D.; Jaglan ,S.; Shankar, R.; Dheer, D.; Shankar ,R.; Arora, D.; Jaglan, S.; Rawal, R. K. Polysaccharides based nanomaterials for targeted anti-cancer drug delivery. Journal of drug targeting ,2017, 25(1), 1-16. |
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143 |
Naseer, S.; Bhat, K. A.; Qadri, M.; Riyaz-Ul-Hassan, S.; Malik, F. A.; Khuroo, M. A. Bioactivity-guided isolation, antimicrobial and cytotoxic evaluation of secondary metabolites from Cladosporium tenuissimum associated with Pinus wallichiana. ChemistrySelect ,2017, 2(3), 1311-1314. |
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144 |
Singh V.; Singh B.; Sharma A.; Kaur K.; Pati P .K.; Gupta A. P.; Salar R. K.; Hallan V. Leaf spot disease adversely affects human health-promoting constituents and withanolide biosynthesis in Withania somnifera (L.) Dunal. Journal of applied microbiology ,2017, 122(1), 153-165. |
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145 |
Dangroo, N.A.; Singh, J.; Gupta, N.; Singh, S.; Kaul, A.; Khuroo, M.A.; Sangwan, P. T- and B-cell immunosuppressive activity of novel alpha-santonin analogs with humoral and cellular immune response in Balb/c mice. Medchemcomm,2017, 8(1), 211-219. |
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146 |
Kumar, B.; Singh, V.; Shankar, R.; Kumar, K.; Rawal, R.K. Synthetic and Medicinal Prospective of Structurally Modified Curcumins. Current Topics in Medicinal Chemistry ,2017, 17(2), 148-161. |
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147 |
Mushtaq, S.; Hassan, Q.P.; Sharma, R.; Majeed, R.; Dar, A.H.; Sultan, P.; Khan, I.A.; Ali, S.A.; Ali, M.N. Evaluation of anticancer and antimicrobial activities of selected medicinal plants of Kashmir Himalayas, India. Indian Journal of Traditional Knowledge, 2017, 16(1), 141-145. |
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148 |
Razdan, S.; Bhat, W.W.; Dhar, N.; Rana, S.; Pandith, S.A.; Wani, T. A.; Vishwakarma, R.; Lattoo, S. K. Molecular characterization of DWF1 from Withania somnifera (L.) Dunal: its implications in withanolide biosynthesis. Journal of Plant Biochemistry and Biotechnology ,2017, 26(1), 52-63. |
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149 |
Mahajan, P.; Suri, N.; Mehra, R.; Gupta, M.; Kumar, A.; Singh, S. K.; Nargotra, A. Discovery of novel small molecule EGFR inhibitory leads by structure and ligand-based virtual screening. Medicinal Chemistry Research ,2017, 26(1), 74-92. |
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150 |
Malik ,T.A.; Kamili ,A. N.; Chishti ,M .Z.; Tantry ,M. A.; Ahad ,S.; Hussain, P. R.; Johri, R .K. Breaking the resistance of Escherichia coli: Antimicrobial activity of Berberis lycium Royle. Microbial pathogenesis , 2017, 10212-20. |
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151 |
Koul, M.; Singh, S. Penicillium spp.: prolific producer for harnessing cytotoxic secondary metabolites. Anti-Cancer Drugs , 2017, 28(1), 11-30. |
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152 |
Lone, M.I.; Nabi, A.; Dar ,N. J.; Hussain, A.; Nazam, N.; Ahmad, W.; Hamid ,A. Toxicogenetic evaluation of dichlorophene in peripheral blood and in the cells of the immune system using molecular and flow cytometric approaches. Chemosphere ,2017, 167520-529. |
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153 |
Rather, G. A.; Sharma, A.; Pandith, S. A.; Kaul, V.; Nandi, U.; Misra, P.; Lattoo, S. K. De novo transcriptome analyses reveals putative pathway genes involved in biosynthesis and regulation of camptothecin in Nothapodytes nimmoniana (Graham) Mabb. Plant Molecular Biology ,2017. |
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154 |
Gupta, S.; Ul Ahsan, A.; Wani, A.; Khajuria, V.; Nazir, L. A.; Sharma, S.; Bhagat, A.; Raj ,S.P.; Bhardwaj, S.; Peerzada, K. J.; et al. The amino analogue of β-boswellic acid efficiently attenuates the release of pro-inflammatory mediators than its parent compound through the suppression of NF-κB/IκBα signalling axis. Cytokine+, 2017, DOI:10.1016/j.cyto.2017.12.004. |
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155 |
Shankar, S.; Faheem, M. M.; Nayak, D.; Wani, N. A.; Farooq, S.; Koul, S.; Goswami, A.; Rai, R. Cyclodipeptide c(Orn-Pro) Conjugate with 4-Ethylpiperic Acid Abrogates Cancer Cell Metastasis through Modulating MDM2. Bioconjugate Chemistry ,2017, DOI:10.1021/acs.bioconjchem.7b00670. |
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156 |
Bhat, Z. S.; Ul Lah, H.; Rather, M.A.; Maqbool, M.; Ara, T.; Ahmad, Z.; Yousuf, S. K. Synthesis and in vitro evaluation of substituted 3-cinnamoyl-4-hydroxy-pyran-2-one (CHP) in pursuit of new potential antituberculosis agents. MedChemComm ,2017, DOI:10.1039/c7md00366h. |
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157 |
Pandey, A. Bani, S.; Dutt, P.; Satti, Naresh .; Avtar, S.K.; Qazi, G. N. Multifunctional neuroprotective effect of Withanone, a compound from Withania somnifera roots in alleviating cognitive dysfunction. Cytokine+, 2017, DOI:10.1016/j.cyto.2017.10.019. |
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158 |
Wani, T. A.; Lattoo, S.K. Auxin response factor (GaARF) cloning and expression in relation to reproductive maturation in Grewia asiatica L. Plant Gene ,2017, 12, 123-130. |
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159 |
Sultan, S.; Gupta, V.; Shah, B. A. Photoredox-Catalyzed Isatin Reactions: Access to Dibenzo-1,7-Naphthyridine Carboxylate and Tryptanthrin. ChemPhotoChem ,2017, 1(4), 120-124. |
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160 |
Arora, D.; Jaglan, S. Therapeutic applications of resveratrol nanoformulations. Environmental Chemistry Letters ,2017, DOI:10.1007/s10311-017-0660-0. |
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161 |
Sharma, A.; Magotra, A.; Rath, S.K.; Wazir, P.; Nandi, U.; Koul, S.; Sangwan, P. L; Gupta, A. P.; Singh, G. In-vitro and in-vivo pharmacokinetics of IS01957, p-coumaric acid derivative using a validated LC-ESI-MS/MS method in mice plasma. Journal of Pharmaceutical Investigation ,2017, DOI:10.1007/s40005-017-0350-8. |
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162 |
Wani, N. A.; Raghothama, S.; Singh, U. P.; Rai, R. C11/C9 Helical folding in αβ hybrid peptides containing 1-amino-cyclohexane acetic acid (β3, 3-Ac6c). Chemistry – A European Journal ,2017, 23(35), 8364-8370. |
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163 |
Dar, N. J.; Satti, N. K.; Dutt, P.; Hamid, A.; Ahmad, M.. Attenuation of Glutamate-Induced Excitotoxicity by Withanolide-A in Neuron-Like Cells: Role for PI3K/Akt/MAPK Signaling Pathway. Molecular Neurobiology ,2017, DOI:10.1007/s12035-017-0515-5. |
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164 |
Vishwakarma, R. Editorial: Medicinal Chemistry Research in India. ACS Medicinal Chemistry Letters ,2017, 8(3), 270-272. |
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165 |
Lone, S. H.; Rehman, S. U.; Bhat, K. A. Synthesis of Gallic-Acid-1-Phenyl-1H-[1,2,3]Triazol-4-yl Methyl Esters as Effective Antioxidants. Drug Research (Stuttgart, Germany) ,2017, 67(2), 111-118. |
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166 |
Arora ,D.; Sharma ,N.; Jaglan, S.; Arora ,D.; Sharma, N.; Chashoo ,G.; Singamaneni, V.; Gupta ,P. Bacillus amyloliquefaciens induces production of a novel blennolide k in co-culture of Setophoma terrestris. Journal of applied microbiology , 2017. |
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167 |
Dheer ,D.; Jyoti; Gupta ,P.N; Shankar, R. Tacrolimus: An updated review on delivering strategies for multifarious diseases. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences ,2017, 114217-227. |
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168 |
Mushtaq, S.; Shah ,A. M.; Shah, A.; Lone, S.A.; Hussain ,A.; Hassan, Q. P.; Ali ,M.N. Bovine mastitis: An appraisal of its alternative herbal cure. Microbial pathogenesis ,2017, 114357-361. |
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169 |
Najar, R.A.; Bhat ,J. A.; Dar ,N. J.; Wani, N. A.; Rahat, B.; Kaur, J.; Gupta, A.P.; Kaur ,J.; Hamid, A. Modulation of dietary folate with age confers selective hepatocellular epigenetic imprints through DNA methylation. The Journal of nutritional biochemistry ,2017, 53121-132. |
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170 |
Singh ,I.; Verma, V.; Chandra ,R.; Singh, I.; Verma ,V.; Singh, S.; Uversky ,V. N.; Uversky ,V.N. In silico evaluation of the resistance of the T790M variant of epidermal growth factor receptor kinase to cancer drug Erlotinib. Journal of biomolecular structure & dynamics ,2017, 1-11. |
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171 |
Magotra ,A.; Sharma, A.; Singh ,S.; Kumar ,S.; Ojha ,P. K.; Bokolia, N.; Khan, I. A.; Wazir, P.; Sharma, S.; Singh, P.P.; et al. Physicochemical, pharmacokinetic, efficacy and toxicity profiling of a potential nitrofuranyl methyl piperazine derivative IIIM-MCD-211 for oral tuberculosis therapy via in-silico-in-vitro-in-vivo approach. Pulmonary pharmacology & therapeutics ,2017. |
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